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 Celiprolol Brand name:- Celipres 100, 200mg tab. Celiprolol is a beta blocker that works specifically on the heart. It works by slowing down the heart rate and makes the heart more efficient at pumping blood around the body. Pharmacodynamic:-  In animals, the β-adrenoceptor blocking activity of celiprolol is more potent than that of sotalol and practolol, and about equipotent with that of propranolol but in man it is about 4 times less potent than atenolol. However, dose-ranging studies employing a range of doses in the same subjects have not been reported and it is possible that celiprolol’s potency has been underestimated. β-Blockade following a single oral dose of 400mg in man can be detected at 24 hours and once-daily dosing is effective in hypertension and angina. Using the standard animal models celiprolol is more selective for the β1- than the β2-adrenoceptor, and in patients with angina the reduction in blood pressure following exercise was larger after treatment with...